Brief Information of the Compound and Protein
Compound Name
1-(3-(pyrrolidine-1-carbonyl)piperidin-1-yl)-2-(1-((1-(4-(trifluoromethyl)phenyl)-1H-pyrrol-3-yl)methyl)piperidin-4-yl)ethanone
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PubChem ID
CID: 45268247
Canonical SMILES
FC(F)(F)c1ccc(cc1)-n1ccc(CN2CCC(CC(=O)N3CCCC(C3)C(=O)N3CCCC3)CC2)c1
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Compound Formula C29H37F3N4O2
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 71 nM
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