Brief Information of the Compound and Protein
Compound Name
 Compound Info 
4-bromo-2-ethyl-5-methyl-N-[3,3,3-trifluoro-2-hydroxy-2-[(1-methyl-3,4-dihydro-2H-naphthalen-1-yl)methyl]propyl]pyrazole-3-carboxamide
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 PubChem ID
CID: 44433485
Canonical SMILES
CCn1nc(C)c(Br)c1C(=O)NCC(O)(CC1(C)CCCc2ccccc12)C(F)(F)F
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Compound Formula C22H27BrF3N3O2
Compound Structure
Protein Name
 Protein Info 
Glucocorticoid receptor
Protein Classification
Transcription factor
>
Nuclear receptor
>
Nuclear hormone receptor subfamily 3
>
Nuclear hormone receptor subfamily 3 group C
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Nuclear hormone receptor subfamily 3 group C member 1
Uniprot ID
P04150
Gene Name
NR3C1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000068 A-549
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 < 1000 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 40.74 nM