Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(piperidin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
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 PubChem ID
CID: 44407664
Canonical SMILES
Clc1ccc(cc1)-c1n(nc2c1ncn(N1CCCCC1)c2=O)-c1ccccc1Cl
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Compound Formula C22H19Cl2N5O
Compound Structure
Protein Name
 Protein Info 
Cannabinoid receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Lipid-like ligand receptor (family A GPCR)
>
Cannabinoid receptor
Uniprot ID
P21554
Gene Name
CNR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
Ki = 20 nM
   TI
   LI
   LO
   TS
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
Ki = 12 nM
   TI
   LI
   LO
   TS