Brief Information of the Compound and Protein
Compound Name
1-[2-[2-[(3S)-3-hydroxypyrrolidin-1-yl]ethyl]indazol-5-yl]-3-(4-phenoxyphenyl)urea
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PubChem ID
CID: 11525369
SID: 16627342
Canonical SMILES
O[C@H]1CCN(CCn2cc3cc(NC(=O)Nc4ccc(Oc5ccccc5)cc4)ccc3n2)C1
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Compound Formula C26H27N5O3
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000863 I3.4.2 Homo sapiens (Human)  1
1
IC50 = 57 nM
   TI
   LI
   LO
   TS