Brief Information of the Compound and Protein
Compound Name
(R)-7-chloro-9-methoxy-1,3,4,10b-tetrahydropyrazino[2,1-a]-isoindol-6(2H)-one
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PubChem ID
CID: 11346775
Canonical SMILES
COc1cc2[C@@H]3CNCCN3C(=O)c2c(Cl)c1
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Compound Formula C12H13ClN2O2
Compound Structure
Protein Name
5-hydroxytryptamine receptor 2A
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P28223
Gene Name
HTR2A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000065 HEK293-EBNA Homo sapiens (Human)  2
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
2
Ki = 4500 nM
   TI
   LI
   LO
   TS