Brief Information of the Compound and Protein
Compound Name
 Compound Info 
3-[1-(1,2-Dihydro-pyridin-2-yl)-1H-indazol-3-yl]-4-[1-(1,4,4a,8a-tetrahydro-naphthalen-2-yl)-1H-indol-3-yl]-pyrrole-2,5-dione
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 PubChem ID
CID: 10188021
SID: 15183509
Canonical SMILES
O=C1NC(=O)C(=C1c1cn(-c2ccc3ccccc3c2)c2ccccc12)c1nn(CCCN2CCCC2)c2ccccc12
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Compound Formula C36H31N5O2
Compound Structure
Protein Name
 Protein Info 
Protein kinase C beta type
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
AGC protein kinase group
>
AGC protein kinase PKC family
>
AGC protein kinase PKC alpha subfamily
Uniprot ID
P05771
Gene Name
PRKCB
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 170 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 44 nM
2 IC50 = 120 nM