Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(R)-N-(1-oxo-1-((3-(1-phenylcyclopropyl)-3H-imidazo[4,5-b]pyridin-2-yl)methylamino)-3-(2,3,6-trifluorophenyl)propan-2-yl)-1-(trifluoromethyl)cyclopropanecarboxamide
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 PubChem ID
CID: 44447296
Canonical SMILES
Fc1ccc(F)c(C[C@@H](NC(=O)C2(CC2)C(F)(F)F)C(=O)NCc2nc3cccnc3n2C2(CC2)c2ccccc2)c1F
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Compound Formula C30H25F6N5O2
Compound Structure
Protein Name
 Protein Info 
Sodium channel protein type 10 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q9Y5Y9
Gene Name
SCN10A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 446 nM
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