Brief Information of the Compound and Protein
Compound Name
3-(4-Ethyl-phenyl)-9-(2,2,2-trifluoro-ethylamino)-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one
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PubChem ID
CID: 11582178
SID: 16684630
Canonical SMILES
CCc1ccc(cc1)-n1cnc2c(sc3nccc(NCC(F)(F)F)c23)c1=O
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Compound Formula C19H15F3N4OS
Compound Structure
Protein Name
Metabotropic glutamate receptor 1
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Small molecule receptor (family C GPCR)
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Neurotransmitter receptor (family C GPCR)
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Metabotropic glutamate receptor
Uniprot ID
Q13255
Gene Name
GRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000094 1321N1 Homo sapiens (Human)  1
1
IC50 = 99 nM
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