Brief Information of the Compound and Protein
Compound Name
N-(2-(2-(1-(3-bromophenyl)ethylidene)hydrazinyl)-2-oxo-1-(4-oxo-3,4-dihydrophthalazin-1-yl)ethyl)benzamide
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PubChem ID
CID: 9589606
SID: 22418887
Canonical SMILES
C/C(=N\NC(=O)C(NC(=O)c1ccccc1)c1n[nH]c(=O)c2ccccc12)c1cccc(Br)c1
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Compound Formula C25H20BrN5O3
Compound Structure
Protein Name
Proteinase-activated receptor 2
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
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Protease-activated receptor
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Protease-activated receptor
Uniprot ID
P55085
Gene Name
F2RL1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  2
1
EC50 = 199.53 nM
   TI
   LI
   LO
   TS
2
EC50 = 200 nM
   TI
   LI
   LO
   TS