Brief Information of the Compound and Protein
Compound Name
(R)-trans-3-{4-[1-(4-tert-Butylcyclohexyl)-3-(3,5-dimethylphenyl)ureidomethyl]benzoylamino}-2-hydroxypropionic acid
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PubChem ID
SID: 56390117
Canonical SMILES
Cc1cc(C)cc(NC(=O)N(Cc2ccc(cc2)C(=O)NC[C@@H](O)C(O)=O)[C@H]2CC[C@@H](CC2)C(C)(C)C)c1
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Compound Formula C30H41N3O5
Compound Structure
Protein Name
Gastric inhibitory polypeptide receptor
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Glucagon-like receptor
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Gastric inhibitory polypeptide receptor
Uniprot ID
P48546
Gene Name
GIPR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000051 BHK-21 Mesocricetus auratus (Golden hamster)  1
1
IC50 = 220 nM
   TI
   LI
   LO
   TS