Brief Information of the Compound and Protein
Compound Name
5-chloro-3-(((1S,3S)-3-(7-methoxy-4-methylquinolin-2-ylamino)cyclohexylamino)methyl)-N,N-dimethyl-1H-indole-1-carboxamide
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PubChem ID
CID: 44442130
Canonical SMILES
COc1ccc2c(C)cc(N[C@H]3CCC[C@@H](C3)NCc3cn(C(=O)N(C)C)c4ccc(Cl)cc34)nc2c1
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Compound Formula C29H34ClN5O2
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 58 nM
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