Brief Information of the Compound and Protein
Compound Name
 Compound Info 
N,15-dimethyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaene-15-carboxamide
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 PubChem ID
CID: 23596254
Canonical SMILES
CN(C(=O)C1(C)CC2c3ccccc3C1c1ccccc21)c1nccs1
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Compound Formula C22H20N2OS
Compound Structure
Protein Name
 Protein Info 
Glucocorticoid receptor
Protein Classification
Transcription factor
>
Nuclear receptor
>
Nuclear hormone receptor subfamily 3
>
Nuclear hormone receptor subfamily 3 group C
>
Nuclear hormone receptor subfamily 3 group C member 1
Uniprot ID
P04150
Gene Name
NR3C1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000068 A-549
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 1236 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 82.5 nM