Brief Information of the Compound and Protein
Compound Name
N-(4-fluorophenyl)-N-methyl-4-oxo-5-[2-[4-(piperidin-1-ylmethyl)phenyl]ethyl]-6,7-dihydropyrazolo[1,5-a]pyrazine-2-carboxamide
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PubChem ID
CID: 44417912
Canonical SMILES
CN(C(=O)c1cc2C(=O)N(CCc3ccc(CN4CCCCC4)cc3)CCn2n1)c1ccc(F)cc1
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Compound Formula C28H32FN5O2
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 5294 nM
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