Brief Information of the Compound and Protein
Compound Name
1-(4-(piperidin-1-ylmethyl)phenethyl)-4-phenethylpiperazin-2-one
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PubChem ID
CID: 44417905
Canonical SMILES
O=C1CN(CCc2ccccc2)CCN1CCc1ccc(CN2CCCCC2)cc1
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Compound Formula C26H35N3O
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 11 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 20 nM
2 Ki = 11 nM