Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(R)-{4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]-6-fluoroquinolin-3-yl}methanol
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 PubChem ID
CID: 16090633
SID: 24736651
Canonical SMILES
C[C@@H]1CN(CCN1C)c1ccc(Nc2c(CO)cnc3ccc(F)cc23)cc1
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Compound Formula C22H25FN4O
Compound Structure
Protein Name
 Protein Info 
Alpha-2C adrenergic receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
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Monoamine receptor
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Adrenergic receptor
Uniprot ID
P18825
Gene Name
ADRA2C
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000796 SC-115
 Cell Line Info 
Mus musculus (Mouse)  1
1
Ki = 38 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 38.02 nM