Brief Information of the Compound and Protein
Compound Name
N-[4-(3,4-dimethylpiperazin-1-yl)phenyl]-2,3,5,8-tetramethylquinolin-4-amine
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PubChem ID
CID: 16090597
SID: 24736610
Canonical SMILES
CC1CN(CCN1C)c1ccc(Nc2c(C)c(C)nc3c(C)ccc(C)c23)cc1
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Compound Formula C25H32N4
Compound Structure
Protein Name
Alpha-2C adrenergic receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
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Monoamine receptor
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Adrenergic receptor
Uniprot ID
P18825
Gene Name
ADRA2C
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000796 SC-115 Mus musculus (Mouse)  1
1
Ki = 390 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 389.94 nM