Brief Information of the Compound and Protein
Compound Name
Biphenyl-2-carboxylic acid [4-(2-oxo-1,2,2a,3,4,5-hexahydro-azepino[4,3,2-cd]indole-6-carbonyl)-phenyl]-amide
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PubChem ID
CID: 9848300
SID: 14810377
Canonical SMILES
O=C(Nc1ccc(cc1)C(=O)N1CCCC2C(=O)Nc3cccc1c23)c1ccccc1-c1ccccc1
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Compound Formula C31H25N3O3
Compound Structure
Protein Name
Vasopressin V2 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Vasopressin and oxytocin receptor
Uniprot ID
P30518
Gene Name
AVPR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 8 nM
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