Brief Information of the Compound and Protein
Compound Name
4-[(2-Fluoro-benzenesulfonylamino)-methyl]-cyclohexanecarboxylic acid (7-methoxy-3a,4,5,9b-tetrahydro-1H-benzo[e]indol-2-yl)-amide
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Canonical SMILES
COc1ccc2C3CC(NC(=O)[C@H]4CC[C@H](CNS(=O)(=O)c5ccccc5F)CC4)=NC3CCc2c1
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Compound Formula C27H32FN3O4S
Compound Structure
Protein Name
Neuropeptide Y receptor type 5
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Neuropeptide Y receptor
Uniprot ID
Q15761
Gene Name
NPY5R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 121 nM
   TI
   LI
   LO
   TS