Brief Information of the Compound and Protein
Compound Name
7-[Bis-(2-methoxy-ethyl)-amino]-3-(2-bromo-4-isopropyl-phenyl)-5-methyl-3H-thiazolo[4,5-d]pyrimidin-2-one
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PubChem ID
CID: 9957428
SID: 14933098
Canonical SMILES
COCCN(CCOC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)sc12
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Compound Formula C21H27BrN4O3S
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 14.5 nM
   TI
   LI
   LO
   TS