Brief Information of the Compound and Protein
Compound Name
9-(2-Bromo-4-isopropyl-phenyl)-6-[ethyl-(2-methoxy-ethyl)-amino]-2,7-dimethyl-7,9-dihydro-purin-8-one
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PubChem ID
CID: 44384780
Canonical SMILES
CCN(CCOC)c1nc(C)nc2n(-c3ccc(cc3Br)C(C)C)c(=O)n(C)c12
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Compound Formula C21H28BrN5O2
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 47.9 nM
   TI
   LI
   LO
   TS