Brief Information of the Compound and Protein
Compound Name
3-[(5-Ethyl-pyrazolo[1,5-a]pyrimidin-7-ylamino)-methyl]-11-(1H-tetrazol-5-yl)-dibenzo[a,d]cyclohepten-5-one
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PubChem ID
CID: 10366402
SID: 15379887
Canonical SMILES
CCc1cc(NCc2ccc3c(cc4ccccc4c(=O)c3c2)-c2nnn[nH]2)n2nccc2n1
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Compound Formula C25H20N8O
Compound Structure
Protein Name
Type-1 angiotensin II receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Angiotensin receptor
Uniprot ID
P30556
Gene Name
AGTR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000880 COS Chlorocebus aethiops (Green monkey)  1
1
Ki = 1.1 nM
   TI
   LI
   LO
   TS